[1]刘万云,霍平,梅光泉,等.橙皮素芳酰腙化合物的微波合成与抑菌活性研究[J].江西师范大学学报(自然科学版),2012,(02):193-195.
 LIU Wan-yun,HUO Ping,MEI Guang-quan,et al.The Study on Microwave Synthesis and Antibacterial Activity of Hesperetin Aromatic Hydrazone Compounds[J].,2012,(02):193-195.
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橙皮素芳酰腙化合物的微波合成与抑菌活性研究()
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《江西师范大学学报》(自然科学版)[ISSN:1006-6977/CN:61-1281/TN]

卷:
期数:
2012年02期
页码:
193-195
栏目:
出版日期:
2012-03-01

文章信息/Info

Title:
The Study on Microwave Synthesis and Antibacterial Activity of Hesperetin Aromatic Hydrazone Compounds
作者:
刘万云;霍平;梅光泉;熊知行;王瑞君
宜春学院江西省高等学校应用化学与化学生物学重点实验室,江西宜春336000;宜春学院江西省天然药物活性成分研究重点实验室,江西宜春336000;宜春学院江西省高等学校应用化学与化学生物学重点实验室,江西宜春,336000
Author(s):
LIU Wan-yun;HUO Ping;MEI Guang-quan;XIONG Zhi-xing;WANG Rui-jun
关键词:
橙皮素酰腙微波合成抑菌活性
Keywords:
hesperetin hydrazone microwave synthesis antibacterial activity
分类号:
O625.43
文献标志码:
A
摘要:
利用微波辐射技术,以橙皮素和芳酰肼为原料设计合成3种橙皮素芳酰腙类化合物,应用红外光谱、核磁共振谱、质谱和元素分析等分析手段对化合物进行了结构表征.抑菌活性实验表明,合成的3种橙皮素芳酰腙类化合物对大肠杆菌、金黄色葡萄球菌和枯草芽孢杆菌的抑菌活性与橙皮素相比均有较大增强.
Abstract:
Three hesperetin aromatic hydrazone compounds are synthesized in good yields under microwave irradiation by reaction of hesperetin with hydrazides. The structures of these compounds are confirmed by IR, 1H NMR, MS spectra and elemental analysis. Inhibition test showed that the hesperetin aromatic hydrazone compounds against Escherichia coli, Staphylococcus aureus and Bacillus subtilis have good antibacterial activity, compared with hesperetin, have a greater enhancement of antibacterial activity.

参考文献/References:

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备注/Memo

备注/Memo:
江西省教育厅科技课题(GJJ09638);江西省天然药物活性成分研究重点实验室开放课题资助项目
更新日期/Last Update: 1900-01-01