参考文献/References:
[1] Narisada M,Yoshida T,Satoh H,et al.Synthetic studies on β-lactam antibiotics.Part 10.Synthesis of 7β-[2-carboxy-2-(4-hydroxyphenyl)acetamido]-7.alpha.-methoxy-3-[[(1-methyl-1H-tetrazol-5-yl)thio]methyl]-1-oxa-1-dethia-3-cephem-4-carboxylic acid disodium salt(6059-S)and its related 1-oxacephems[J].J Med Chem,1979,22(7):757-759.
[2] Madauss K P,Stewart E L,Williams S P.The evolution of progesterone receptor ligands[J].Medicinal Research Reviews,2007,27(3):374-400.
[3] Bollo S,Nún～ez-Vergara L J,Kang S,et al.The effect of 5-substitution on the electrochemical behavior and antitubercular activity of PA-824[J].Bioorganic and Medicinal Chemistry Letters,2011,21(2):812-817.
[4] Pham V C,Jossang A,Sevenet T,et al.Myrioneurinol:a novel alkaloid skeleton from Myrioneuron nutans[J].Tetrahedron,2007,63(46):11244-11249.
[5] Cocuzza A J,Chidester D R,Cordova B C,et al.Synthesis and evaluation of efavirenz(SustivaTM)analogues as HIV-1 reverse transcriptase inhibitors:replacement of the cyclopropylacetylene side chain[J].Bioorganic and Medicinal Chemistry Letters,2001,11(9):1177-1179.
[6] Liu Haifeng,Ji Min,Cai Jin.Short and efficient approach towards buxozine-C,an alkaloid from Buxus sempervirens[J].Archiv der Pharmazie:An International Journal Pharmaceutical and Medicinal Chemistry,2006,339(12):675-676.
[7] Butler J D,Solano D M,Robins L I,et al.A facile synthesis of new 5H-indazolo[3,2-b] benzo[d]-1,3-oxazines via one-pot intramolecular bis-heterocyclizations[J].The Journal of Organic Chemistry,2008,73(1):234-240.
[8] Vrouenraets S M E,Wit F W N M,Tongeren J,et al.Efavirenz: a review[J].Expert Opinion on Pharmacotherapy,2007,8(6):851-871.
[9] Csütörtöki R,Szatmári I,Koch A,et al.Synthesis and conformational analysis of new naphth[1,2-e][1,3] oxazino[3,4-c] quinazoline derivatives[J].Tetrahedron,2011,67(44):8564-8571.
[10] Avila B,Solano D M,Haddadin M J,et al.Facile syntheses of novel benzo-1,3-dioxolo-,benzothiazolo-,pyrido-,and quinolino-fused 5H-benzo[d]-pyrazolo[5,1-b][1,3]-oxazines and 1H-pyrazoles[J].Organic Letters,2011,13(5):1060-1063.
[11] Asghari S,Habibi A K.One pot three-component regioselective and diastereoselective synthesis of halogenated pyrido[2,1-b][1,3] oxazines[J].Tetrahedron,2012,68(43):8890-8898.
[12] Grigg R D,Schomaker J M,Timokhin V.C-H amination/cyclocarbonylation of allene carbamates:a versatile platform for the synthesis of α,β-unsaturated γ-lactams[J].Tetrahedron,2011,67(24):4318-4326.
[13] Jakobsen P,Horneman A M,Persson E.Inhibitors of the tissue factor/factor VIIa-induced coagulation:synthesis and in vitro evaluation of novel 2-aryl substituted pyrido[3,4-d][1,3]-,pyrido[2,3-d][1,3]-,pyrazino[2,3-d][1,3]-,pyrimido[4,5-d][1,3]-,pyrazolo[3,4-d][1,3]-,thieno[3,2-d][1,3]- and thieno[2,3-d][1,3]-oxazin-4-ones[J].Bioorganic and Medicinal Chemistry,2000,8(12):2803-2812.
[14] Omran O A,Sayed S M,Raslan M A.Iminophosphoranes in heterocyclic synthesis:a facile synthesis of pyrido[4,3-d] pyrimidine and pyrido[4,3-d][1,3] oxazine derivatives via intermolecular aza-wittig reactions[J].Journal of Heterocyclic Chemistry,2017,54(2):1103-1108.
[15] Mo Wenyan,Liang Yonggu,He Hongwu,et al.Facile synthesis and biological activities of novel fluorine-containing pyrido[4,3-d]pyrimidines[J].Journal of Fluorine Chemistry,2008,129(6):519-523.
[16] Mo Wenyan,Liang Yonggu,He Hongwu,et al.Synthesis and cytotoxicity of 8-cyano-3-substitutedalkyl-5-methyl-4-methylene-7-methoxy-3,4-dihydropyrido[4,3-d]pyrimidines[J].Bioorg Med Chem Lett,2011,21(19):5975-5977.
[17] 丁明武.杂环合成中的维悌希反应[M].武汉:华中师范大学出版社,1997.
[18] 王涛.靶标酶抑制剂的设计、合成与性质研究[D].武汉:华中师范大学,2004.
[19] 赵安林,王涛,罗劲,等.新型2-烷硫基-噻吩并[2,3-d]嘧啶-4-酮衍生物的设计、合成与除草活性[J].有机化学,2017,37(7):1877-1882.
[20] 王涛,罗劲,郑彩华.3,6-二烷硫基-1-苯基-吡唑并[3,4-d]嘧啶-4-酮衍生物的合成与除草活性[J].有机化学,2010,30(11):1749-1753.